| Nomenclature | PLD1 | PLD2 |
| HGNC, UniProt | PLD1, Q13393 | PLD2, O14939 |
| EC number | 3.1.4.4 | 3.1.4.4 A phosphatidylcholine + H2O <=> choline + a phosphatidate |
| Endogenous activators | ADP‐ribosylation factor 1 (ARF1, P84077), PIP2, RhoA, PKC evoked phosphorylation, RalA [201, 323] | ADP‐ribosylation factor 1 (ARF1, P84077), PIP2 [316], oleic acid [454] |
| Endogenous inhibitors | Gβ γ [418] | Gβ γ [418] |
| Inhibitors | FIPI (pIC50 8) [463] | FIPI (pIC50 7.8) [484] |
| Selective inhibitors | compound 69 (pIC50 7.3) [463] | VU0364739 (pIC50 7.7) [293] |