| Nomenclature | mechanistic target of rapamycin |
| HGNC, UniProt | MTOR, P42345 |
| EC number | 2.7.11.1 |
| Common abreviation | mTOR |
| Inhibitors | ridaforolimus (pIC50 9.7) [441], torin 1 (pIC50 9.5) [310], INK‐128 (pIC50 9) [231], INK‐128 (pK i 8.9) [231], gedatolisib (pIC50 8.8) [544], dactolisib (pIC50 8.2) [332], PP‐242 (pIC50 8.1) [15], PP121 (pIC50 8) [15], XL388 (pIC50 8) [511], PF‐04691502 (pK i 7.8) [309], apitolisib (pK i 7.8) [506] |
| Selective inhibitors | everolimus (pIC50 8.7) [464], temsirolimus (pIC50 5.8) [278] |