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. Author manuscript; available in PMC: 2014 Jan 28.
Published in final edited form as: J Chem Inf Model. 2012 Dec 28;53(1):230–240. doi: 10.1021/ci300510n

Table 6.

Performance of different FINDSITE based methods for the 168 Human GPCRs

Method (binding database) Average EF0.01 # (%) of targets having EF0.01 > 1
FINDSITE (PDB) 7.1 35 (21%)
FINDSITEX (DrugBank) 10.1 76 (45%)
FINDSITEX (ChEMBL) 19.9 105 (63%)
FINDSITEfilt (PDB)3 8.5 54 (32%)
FINDSITEcomb 22.3 113 (67%)