Table 6.
Performance of different FINDSITE based methods for the 168 Human GPCRs
| Method (binding database) | Average EF0.01 | # (%) of targets having EF0.01 > 1 |
|---|---|---|
| FINDSITE (PDB) | 7.1 | 35 (21%) |
| FINDSITEX (DrugBank) | 10.1 | 76 (45%) |
| FINDSITEX (ChEMBL) | 19.9 | 105 (63%) |
| FINDSITEfilt (PDB)3 | 8.5 | 54 (32%) |
| FINDSITEcomb | 22.3 | 113 (67%) |