Table 2.
S1P4-R agonist activity of 13a–13f
![]() 13a–f | ||
|---|---|---|
| cpd | L | EC50 (nM)α |
| 13a |
|
NA |
| 13b |
|
920 |
| 13c |
|
NA |
| 13d |
|
NA |
| 13e |
|
NA |
| 13f |
|
NA |
Data are reported as mean of n = 3 determinations. NA = not active at concentrations up to 25 μM.
S1P4-R agonist activity of 13a–13f
![]() 13a–f | ||
|---|---|---|
| cpd | L | EC50 (nM)α |
| 13a |
|
NA |
| 13b |
|
920 |
| 13c |
|
NA |
| 13d |
|
NA |
| 13e |
|
NA |
| 13f |
|
NA |
Data are reported as mean of n = 3 determinations. NA = not active at concentrations up to 25 μM.