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. 2024 Nov 5;31(12):1884–1894. doi: 10.1038/s41417-024-00847-8

Table 3.

Pharmacokinetic parameters of S2172.

Cmax (µM) 1.20 ± 0.12
Tmax (hr) 0.25
T1/2 (hr) 4.98 ± 1.64
AUC0–6 h (µM·hr) 1.11 ± 0.08
Plasma concentration at 0.5 hr (µM) 0.75 ± 0.09
Brain concentration at 0.5 hr (µM) 1.52 ± 0.14
Brain/plasma ratio 2.06 ± 0.39

Pharmacokinetic parameters were determined in 8-week-old Crl:CD1 (ICR) mice treated with a single intraperitoneal injection at 30 mg/kg (n = 3).